Active Ingredient Sirolimus

Active Ingredient Details

What is Sirolimus?

A macrolide compound obtained from Streptomyces hygroscopicus that acts by selectively blocking the transcriptional activation of cytokines thereby inhibiting cytokine production. It is bioactive only when bound to IMMUNOPHILINS. Sirolimus is a potent immunosuppressant and possesses both antifungal and antineoplastic properties.

What is the usage for Sirolimus?

Sirolimus is used with other medications to prevent rejection of a kidney transplant. This medication belongs to a class of drugs known as immunosuppressants. It works by weakening your body's defense system (immune system) to help your body accept the new organ as if it were your own. Sirolimus may also be used to treat a certain lung disease (lymphangioleiomyomatosis-LAM).

How many products in the NDC database contain Sirolimus?

The NDC database has 59 products with the active ingredient Sirolimus. The following table lists all the products that have this active ingredient.

NDC Products with Sirolimus

NDC Proprietary Name Non-Proprietary Name Dosage Form Route Name Company Name Status
0008-1041Proprietary Name: Rapamune SirolimusTablet, Sugar CoatedOralWyeth Pharmaceuticals Llc, A Subsidiary Of Pfizer Inc.ACTIVE
0008-1042Proprietary Name: Rapamune SirolimusTablet, Sugar CoatedOralWyeth Pharmaceuticals Llc, A Subsidiary Of Pfizer Inc.ACTIVE
0904-7248Proprietary Name: Sirolimus SirolimusTabletOralMajor PharmaceuticalsACTIVE
16714-187Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralNorthstar Rx LlcACTIVE
16714-188Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralNorthstar Rx LlcACTIVE
16714-189Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralNorthstar Rx LlcACTIVE
31722-316Proprietary Name: Sirolimus SirolimusSolutionOralCamber Pharmaceuticals, Inc.ACTIVE
42513-0013Proprietary Name: SirolimusPowderLivzon Group Fuzhou Fuxing Pharmaceutical Co., Ltd.ACTIVE
42816-1040Proprietary Name: SirolimusTablet, Sugar CoatedPfizer Ireland Pharmaceuticals Unlimited CompanyACTIVE
42816-1041Proprietary Name: SirolimusTablet, Sugar CoatedPfizer Ireland Pharmaceuticals Unlimited CompanyACTIVE
42816-1042Proprietary Name: SirolimusTablet, Sugar CoatedPfizer Ireland Pharmaceuticals Unlimited CompanyACTIVE
49187-0801Proprietary Name: RapamycinPowderLonza AgACTIVE
50268-718Proprietary Name: Sirolimus SirolimusTabletOralAvpakACTIVE
51187-0010Proprietary Name: SirolimusPowderHisun Pharmaceutical (hangzhou) Co., Ltd.ACTIVE
52076-6216Proprietary Name: RapamycinPowderChunghwa Chemical Synthesis & Biotech. LtdACTIVE
55111-653Proprietary Name: Sirolimus SirolimusTabletOralDr. Reddy's Laboratories LimitedACTIVE
55111-654Proprietary Name: Sirolimus SirolimusTabletOralDr. Reddy's Laboratories LimitedACTIVE
55486-1571Proprietary Name: SirolimusPowderCuria Italy S.r.l.ACTIVE
55486-1592Proprietary Name: Sirolimus ComplexPowderCuria Italy S.r.l.ACTIVE
55500-0011Proprietary Name: SirolimusPowderNorth China Pharmaceutical Huasheng Co. Ltd.ACTIVE
56125-800Proprietary Name: SirolimusSuspensionNovo Nordisk Production Ireland LimitedACTIVE
57885-0014Proprietary Name: SirolimusPowderChongqing Daxin Pharmaceutical Co. Ltd.ACTIVE
59573-0004Proprietary Name: SirolimusPowderFujian Kerui Pharmaceutical Co., Ltd.ACTIVE
59762-1001Proprietary Name: Sirolimus SirolimusTablet, Sugar CoatedOralMylan Pharmaceuticals Inc.ACTIVE
59762-1002Proprietary Name: Sirolimus SirolimusTablet, Sugar CoatedOralMylan Pharmaceuticals Inc.ACTIVE
59762-1003Proprietary Name: Sirolimus SirolimusTablet, Sugar CoatedOralMylan Pharmaceuticals Inc.ACTIVE
59762-1205Proprietary Name: Sirolimus SirolimusSolutionOralMylan Pharmaceuticals Inc.ACTIVE
60505-6197Proprietary Name: Sirolimus SirolimusSolutionOralApotex CorpACTIVE
62991-3184Proprietary Name: SirolimusPowderLetco Medical, LlcACTIVE
65727-013Proprietary Name: SirolimusPowderBiocon LimitedACTIVE
65841-771Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralZydus Lifesciences LimitedACTIVE
65841-772Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralZydus Lifesciences LimitedACTIVE
65841-773Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralZydus Lifesciences LimitedACTIVE
66689-347Proprietary Name: Sirolimus SirolimusSolutionOralVistapharm, LlcACTIVE
67877-746Proprietary Name: Sirolimus SirolimusTabletOralAscend Laboratories, LlcACTIVE
67877-747Proprietary Name: Sirolimus SirolimusTabletOralAscend Laboratories, LlcACTIVE
67877-748Proprietary Name: Sirolimus SirolimusTabletOralAscend Laboratories, LlcACTIVE
68084-915Proprietary Name: Sirolimus SirolimusTabletOralAmerican Health PackagingACTIVE
68254-1006Proprietary Name: SirolimusPowderConcord Biotech LtdACTIVE
68382-351Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralZydus Pharmaceuticals Usa Inc.ACTIVE
68382-352Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralZydus Pharmaceuticals Usa Inc.ACTIVE
68382-520Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralZydus Pharmaceuticals Usa Inc.ACTIVE
68462-682Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralGlenmark Pharmaceuticals Inc., UsaACTIVE
68462-683Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralGlenmark Pharmaceuticals Inc., UsaACTIVE
68462-684Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralGlenmark Pharmaceuticals Inc., UsaACTIVE
69238-1594Proprietary Name: Sirolimus SirolimusSolutionOralAmneal Pharmaceuticals Ny LlcACTIVE
70518-3546Proprietary Name: Sirolimus SirolimusTabletOralRemedyrepack Inc.ACTIVE
70518-4194Proprietary Name: Sirolimus SirolimusTablet, Sugar CoatedOralRemedyrepack Inc.ACTIVE
70518-4376Proprietary Name: Sirolimus SirolimusTablet, Film CoatedOralRemedyrepack Inc.ACTIVE
71052-202Proprietary Name: SirolimusPowderDarmerica, LlcACTIVE
72205-099Proprietary Name: Sirolimus SirolimusSolutionOralNovadoz Pharmaceuticals LlcACTIVE
73212-019Proprietary Name: SirolimusPowderQingdao Biopeptek Co., Ltd.ACTIVE
73377-024Proprietary Name: SirolimusPowderAx Pharmaceutical CorpACTIVE
73683-101Proprietary Name: Hyftor SirolimusGelTopicalNobelpharma America, LlcACTIVE
80803-153Proprietary Name: Fyarro SirolimusInjection, Powder, Lyophilized, For SuspensionIntravenousAadi BioscienceACTIVE
82393-501Proprietary Name: Sirolimus (rapamycin)PowderPharma Source Direct, Inc.ACTIVE
84517-032Proprietary Name: SirolimusPowderZhejiang Wild Wind Pharmaceutical Co.,ltd.ACTIVE
85512-2027Proprietary Name: SirolimusPowderQingdao Qinzeyuan Biotechnology Co., LtdACTIVE
85705-001Proprietary Name: SirolimusPowderSumar Biotech LlpACTIVE
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