Cytochrome P450 3A5 Inhibitors [MoA] - N0000190115

Pharmacologic Class Information

Pharmacologic Code N0000190115
Pharmacologic Name Cytochrome P450 3A5 Inhibitors
Pharmacologic Uses
  • azole antifungal
  • cortisol synthesis inhibitor
  • hepatitis C virus (HCV) NS3/4A protease inhibitor
  • nitroimidazole antimicrobial
Pharmacologic Concept Mechanisms of Action - [MoA]
Pharmacologic Concept Description This concept refers to the mechanism of action pharmacologic action at the receptor, membrane, or tissue level. In MED-RT, molecular, subcellular, or cellular effects of drug generic ingredients, organized into a chemical function classification hierarchy, beneath the "Cellular or Molecular Interactions" concept.

NDC Products with Cytochrome P450 3A5 Inhibitors

The table contains 79 products whose active ingredient are classified under the same pharmacologic class Cytochrome P450 3A5 Inhibitors [MoA].

NDC Proprietary Name Non-Proprietary Name Dosage Form Route Name Company Name Status
0024-4512Fexinidazole Non-Proprietary Name: FexinidazoleTabletOralSanofi-aventis U.s. LlcACTIVE
0093-3219Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalTeva Pharmaceuticals Usa, Inc.ACTIVE
0168-0099Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalE. Fougera & Co. A Division Of Fougera Pharmaceuticals Inc.ACTIVE
0713-0592Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalCosette Pharmaceuticals, Inc.ACTIVE
16714-955Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalNorthstar Rx LlcACTIVE
21922-025Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalEncube Ethicals Private LimitedACTIVE
35573-433Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralBurel Pharmaceuticals, LlcACTIVE
43538-530Ketodan Non-Proprietary Name: KetoconazoleAerosol, FoamTopicalMedimetriks Pharmaceuticals, Inc.ACTIVE
45802-465Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalPadagis Israel Pharmaceuticals LtdACTIVE
45802-532Ketoconazole Non-Proprietary Name: KetoconazoleAerosol, FoamTopicalPadagis Israel Pharmaceuticals LtdACTIVE
50090-3288Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalA-s Medication SolutionsACTIVE
50090-5265Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalA-s Medication SolutionsACTIVE
50090-6046Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalA-s Medication SolutionsACTIVE
50090-6069Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalA-s Medication SolutionsACTIVE
50090-6142Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralA-s Medication SolutionsACTIVE
50090-7538Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalA-s Medication SolutionsACTIVE
51407-279Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalGolden State Medical Supply, Inc.ACTIVE
51672-1298Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalSun Pharmaceutical Industries, Inc.ACTIVE
51672-4026Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralTaro Pharmaceuticals U.s.a., Inc.ACTIVE
55292-320Isturisa Non-Proprietary Name: OsilodrostatTablet, CoatedOralRecordati Rare Diseases, Inc.ACTIVE
55292-321Isturisa Non-Proprietary Name: OsilodrostatTablet, CoatedOralRecordati Rare Diseases, Inc.ACTIVE
55292-330Isturisa Non-Proprietary Name: OsilodrostatTablet, CoatedOralRecordati Rare Diseases, Inc.ACTIVE
55292-331Isturisa Non-Proprietary Name: OsilodrostatTablet, CoatedOralRecordati Rare Diseases, Inc.ACTIVE
55505-192Nizoral Non-Proprietary Name: KetoconazoleShampooTopicalKramer LaboratoriesACTIVE
55505-196Nizoral Non-Proprietary Name: KetoconazoleShampooTopicalKramer LaboratoriesACTIVE
55505-233Nizoral Non-Proprietary Name: KetoconazoleShampooTopicalKramer LaboratoriesACTIVE
60429-020Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralGolden State Medical Supply, Inc.ACTIVE
63187-774Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalProficient Rx LpACTIVE
63629-8675Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalBryant Ranch PrepackACTIVE
63629-8676Ketoconazole Non-Proprietary Name: KetoconazoleAerosol, FoamTopicalBryant Ranch PrepackACTIVE
63629-8677Ketoconazole Non-Proprietary Name: KetoconazoleAerosol, FoamTopicalBryant Ranch PrepackACTIVE
63629-8819Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalBryant Ranch PrepackACTIVE
63629-8820Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalBryant Ranch PrepackACTIVE
63646-010Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalTolmar Inc.ACTIVE
64380-827Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralStrides Pharma Science LimitedACTIVE
67296-0448Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalRedpharm DrugACTIVE
67296-0540Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalRedpharm DrugACTIVE
67296-1807Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalRedpharm DrugACTIVE
67296-2089Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalRedpharm DrugACTIVE
68071-1709Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalNucare Pharmaceuticals,inc.ACTIVE
68071-3512Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalNucare Pharmaceuticals,inc.ACTIVE
68788-8233Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalPreferred Pharmaceuticals Inc.ACTIVE
68788-8257Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalPreferred Pharmaceuticals Inc.ACTIVE
68788-8868Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalPreferred Pharmaceuticals Inc.ACTIVE
69292-224Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralAmici Pharma Inc.ACTIVE
70518-4236Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalRemedyrepack Inc.ACTIVE
70700-160Ketoconazole Non-Proprietary Name: Ketoconazole FoamAerosol, FoamTopicalXiromed, LlcACTIVE
70771-1874Ketoconazole Non-Proprietary Name: KetoconazoleShampooTopicalZydus Lifesciences LimitedACTIVE
70954-662Ketoconazole Non-Proprietary Name: KetoconazoleSuspensionTopicalAni Pharmaceuticals, Inc.ACTIVE
71085-008Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalIpg Pharmaceuticals, Inc.ACTIVE
71205-105Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalProficient Rx LpACTIVE
71335-0439Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralBryant Ranch PrepackACTIVE
71335-1849Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralBryant Ranch PrepackACTIVE
71713-097Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalThirty Madison IncACTIVE
72162-1409Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalBryant Ranch PrepackACTIVE
72162-1417Ketoconazole Non-Proprietary Name: KetoconazoleAerosol, FoamTopicalBryant Ranch PrepackACTIVE
72189-180Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralDirect RxACTIVE
72189-422Ketoconazole Cream Non-Proprietary Name: Ketoconazole CreamCreamTopicalDirect_rxACTIVE
72189-428Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralDirect_rxACTIVE
72578-156Ketoconazole Non-Proprietary Name: KetoconazoleShampooTopicalViona Pharmaceuticals IncACTIVE
72789-052Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralPd-rx Pharmaceuticals, Inc.ACTIVE
82804-091Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalProficient Rx LpACTIVE
83364-005Fungifree Nail Fungus Treatment Non-Proprietary Name: Ketoconazole, TolnaftateSolutionTopicalYitongbada (shenzhen) International Trade Co., LtdACTIVE
83887-004Pureskin Scalp Protection Anti Dandruff Shampoo. Non-Proprietary Name: Pureskin Scalp Protection Anti Dandruff ShampooShampooTopicalChangsha Beiliang E-commerce Co., LtdACTIVE
83887-005Derphea Advanced Scalp Shampoo. Non-Proprietary Name: Advanced Scalp ShampooShampooTopicalChangsha Beiliang E-commerce Co., LtdACTIVE
84277-5665Danil Non-Proprietary Name: Danil Compound Ketoconazole Solution For Scalp Disorders.SolutionTopicalJiangsu Chenpai Bond Pharmaceutical Co.,ltd.ACTIVE
84277-5666Danil Non-Proprietary Name: Danil Compound Ketoconazole Solution For Scalp Disorders.LotionTopicalJiangsu Chenpai Bond Pharmaceutical Co.,ltd.ACTIVE
84372-037Lanimpress1%ketoconazoleantidandruffshampoo Non-Proprietary Name: Lanimpress1%ketoconazoleantidandruffshampooLotionTopicalShenzhen Zhumeng Times Technology Co., Ltd.ACTIVE
84372-038Lanimpress1%ketoconazoleantidandruffshampoo Non-Proprietary Name: Lanimpress1%ketoconazoleantidandruffshampooLotionTopicalShenzhen Zhumeng Times Technology Co., Ltd.ACTIVE
84372-039Lanimpress1%ketoconazoleantidandruffshampoo Non-Proprietary Name: Lanimpress1%ketoconazoleantidandruffshampooLotionTopicalShenzhen Zhumeng Times Technology Co., Ltd.ACTIVE
84372-040Lanimpress1%ketoconazoleantidandruffshampoo Non-Proprietary Name: Lanimpress1%ketoconazoleantidandruffshampooLotionTopicalShenzhen Zhumeng Times Technology Co., Ltd.ACTIVE
84372-041Lanimpress1%ketoconazoleantidandruffshampoo Non-Proprietary Name: Lanimpress1%ketoconazoleantidandruffshampooLotionTopicalShenzhen Zhumeng Times Technology Co., Ltd.ACTIVE
84372-042Lanimpress1%ketoconazoleantidandruffshampoo Non-Proprietary Name: Lanimpress1%ketoconazoleantidandruffshampooLotionTopicalShenzhen Zhumeng Times Technology Co., Ltd.ACTIVE
84558-0051% Ketoconazole Anti Dandruff Non-Proprietary Name: 1% Ketoconazole Anti Dandruff ShampooShampooCutaneousGuangzhou Yusong Fine Chemicls Co., LtdACTIVE
84659-9040Vixa Skineal Non-Proprietary Name: Vixa Skineal Compound KetoconazoleCreamTopicalYunnan Yuyao Bio-pharmaceutical Co.,ltd.ACTIVE
84745-002Poagci Ketoconazole Vcp-kad001 Non-Proprietary Name: KetoconazoleLiquidTopicalVince (guangzhou) Cosmetics Co., Ltd.ACTIVE
85384-00011% Ketoconazole Non-Proprietary Name: KetoconazoleShampooTopicalTagrid LlcACTIVE
85384-0002Tagrit Antifungal Treament Ketoconazole 1% Non-Proprietary Name: KetoconazoleCreamTopicalTagrid LlcACTIVE
85521-001Dandrx 1% Ketoconazole Anti-dandruff Non-Proprietary Name: Dandrx 1% Ketoconazole Anti-dandruff ShampooLiquidTopicalDandrx LlcACTIVE