Cytochrome P450 3A5 Inhibitors [MoA] - N0000190115

Pharmacologic Class Information

Pharmacologic Code N0000190115
Pharmacologic Name Cytochrome P450 3A5 Inhibitors
Pharmacologic Uses
  • azole antifungal
  • cortisol synthesis inhibitor
  • hepatitis C virus (HCV) NS3/4A protease inhibitor
  • nitroimidazole antimicrobial
Pharmacologic Concept Mechanisms of Action - [MoA]
Pharmacologic Concept Description This concept refers to the mechanism of action pharmacologic action at the receptor, membrane, or tissue level. In MED-RT, molecular, subcellular, or cellular effects of drug generic ingredients, organized into a chemical function classification hierarchy, beneath the "Cellular or Molecular Interactions" concept.

NDC Products with Cytochrome P450 3A5 Inhibitors

The table contains 58 products whose active ingredient are classified under the same pharmacologic class Cytochrome P450 3A5 Inhibitors [MoA].

NDC Proprietary Name Non-Proprietary Name Dosage Form Route Name Company Name Status
0024-4512Fexinidazole Non-Proprietary Name: FexinidazoleTabletOralSanofi-aventis U.s. LlcACTIVE
0093-3219Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalTeva Pharmaceuticals Usa, Inc.ACTIVE
0168-0099Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalE. Fougera & Co. A Division Of Fougera Pharmaceuticals Inc.ACTIVE
0186-0776Brilinta Non-Proprietary Name: TicagrelorTabletOralAstrazeneca Pharmaceuticals LpACTIVE
0186-0777Brilinta Non-Proprietary Name: TicagrelorTabletOralAstrazeneca Pharmaceuticals LpACTIVE
0378-7007Ketaconazole Non-Proprietary Name: KetaconazoleAerosol, FoamTopicalMylan Pharmaceuticals Inc.ACTIVE
16714-955Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalNorthstar Rx LlcACTIVE
21922-025Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalEncube Ethicals Private LimitedACTIVE
35573-433Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralBurel Pharmaceuticals, LlcACTIVE
43538-530Ketodan Non-Proprietary Name: KetoconazoleAerosol, FoamTopicalMedimetriks Pharmaceuticals, Inc.ACTIVE
45802-465Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalPadagis Israel Pharmaceuticals LtdACTIVE
45802-532Ketoconazole Non-Proprietary Name: KetoconazoleAerosol, FoamTopicalPadagis Israel Pharmaceuticals LtdACTIVE
50090-0720Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalA-s Medication SolutionsACTIVE
50090-5265Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalA-s Medication SolutionsACTIVE
50090-6046Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalA-s Medication SolutionsACTIVE
50090-6069Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalA-s Medication SolutionsACTIVE
50090-6142Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralA-s Medication SolutionsACTIVE
51407-279Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalGolden State Medical Supply, Inc.ACTIVE
51672-1298Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalTaro Pharmaceuticals U.s.a., Inc.ACTIVE
51672-4026Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralTaro Pharmaceuticals U.s.a., Inc.ACTIVE
55154-9618Brilinta Non-Proprietary Name: TicagrelorTabletOralCardinal Health 107, LlcACTIVE
55292-320Isturisa Non-Proprietary Name: OsilodrostatTablet, CoatedOralRecordati Rare Diseases, Inc.ACTIVE
55292-321Isturisa Non-Proprietary Name: OsilodrostatTablet, CoatedOralRecordati Rare Diseases, Inc.ACTIVE
55292-322Isturisa Non-Proprietary Name: OsilodrostatTablet, CoatedOralRecordati Rare Diseases, Inc.ACTIVE
55505-192Nizoral Non-Proprietary Name: KetoconazoleShampooTopicalKramer LaboratoriesACTIVE
55505-196Nizoral Non-Proprietary Name: KetoconazoleShampooTopicalKramer LaboratoriesACTIVE
60429-020Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralGolden State Medical Supply Inc.ACTIVE
63187-774Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalProficient Rx LpACTIVE
63629-8675Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalBryant Ranch PrepackACTIVE
63629-8676Ketoconazole Non-Proprietary Name: KetoconazoleAerosol, FoamTopicalBryant Ranch PrepackACTIVE
63629-8677Ketoconazole Non-Proprietary Name: KetoconazoleAerosol, FoamTopicalBryant Ranch PrepackACTIVE
63629-8819Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalBryant Ranch PrepackACTIVE
63629-8820Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalBryant Ranch PrepackACTIVE
63646-010Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalTolmar Inc.ACTIVE
64380-827Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralStrides Pharma Science LimitedACTIVE
66267-400Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralNucare Pharmaceuticals,inc.ACTIVE
68071-2309Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalNucare Pharmaceuticals,inc.ACTIVE
68071-2847Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalNucare Pharmaceuticals,inc.ACTIVE
68071-2902Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralNucare Pharmaceuticals,inc.ACTIVE
68788-7755Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalPreferred Pharmaceuticals, Inc.ACTIVE
68788-8233Ketoconazole Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalPreferred Pharmaceuticals Inc.ACTIVE
68788-8257Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalPreferred Pharmaceuticals Inc.ACTIVE
68788-9903Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalPreferred Pharmaceuticals, Inc.ACTIVE
68788-9915Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalPreferred Pharmaceuticals, Inc.ACTIVE
69238-1134Ticagrelor Non-Proprietary Name: TicagrelorTabletOralAmneal Pharmaceuticals Ny LlcACTIVE
70518-0915Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralRemedyrepack Inc.ACTIVE
70518-2831Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralRemedyrepack Inc.ACTIVE
70518-3367Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalRemedyrepack Inc.ACTIVE
70700-160Ketoconazole Non-Proprietary Name: Ketoconazole FoamAerosol, FoamTopicalXiromed, LlcACTIVE
71085-008Ketoconazole Non-Proprietary Name: KetoconazoleCreamTopicalIpg Pharmaceuticals, Inc.ACTIVE
71205-105Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalProficient Rx LpACTIVE
71335-1849Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralBryant Ranch PrepackACTIVE
71713-097Ketoconazole Non-Proprietary Name: KetoconazoleShampoo, SuspensionTopicalThirty Madison IncACTIVE
72189-180Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralDirect RxACTIVE
72189-422Ketoconazole Cream Non-Proprietary Name: Ketoconazole CreamCreamTopicalDirect_rxACTIVE
72189-428Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralDirect_rxACTIVE
72641-005Ketoconazole Cream, 2% Non-Proprietary Name: Ketoconazole Cream, 2%CreamTopicalTasman Pharma Inc.ACTIVE
72789-052Ketoconazole Non-Proprietary Name: KetoconazoleTabletOralPd-rx Pharmaceuticals, Inc.ACTIVE