Breast Cancer Resistance Protein Inhibitors [MoA] - N0000190113

Pharmacologic Class Information

Pharmacologic Code N0000190113
Pharmacologic Name Breast Cancer Resistance Protein Inhibitors
Pharmacologic Uses
  • azole antifungal
  • CYP3A inhibitor
  • cytomegalovirus (CMV) pUL97 kinase inhibitor
  • endothelin and angiotensin II receptor antagonist
  • estrogen receptor antagonist
  • farnesyltransferase inhibitor
  • gonadotropin-releasing hormone (GnRH) receptor antagonist
  • hepatitis C virus (HCV) NS3/4A protease inhibitor
  • hepatitis C virus (HCV) NS5A inhibitor
  • hepatitis C virus non-nucleoside NS5B palm polymerase inhibitor
  • HIV-1 protease inhibitor
  • human immunodeficiency virus type 1 (HIV-1) capsid inhibitor
  • inhibitor of the orthopoxvirus VP37 envelope wrapping protein
  • kinase inhibitor
  • monoamine oxidase type B (MAO-B) inhibitor
  • oxazolidinone antibacterial
  • phenylalanine hydroxylase activator
  • substance P/neurokinin-1 (NK-1) receptor antagonist
  • thrombopoietin receptor agonist
Pharmacologic Concept Mechanisms of Action - [MoA]
Pharmacologic Concept Description This concept refers to the mechanism of action pharmacologic action at the receptor, membrane, or tissue level. In MED-RT, molecular, subcellular, or cellular effects of drug generic ingredients, organized into a chemical function classification hierarchy, beneath the "Cellular or Molecular Interactions" concept.

NDC Products with Breast Cancer Resistance Protein Inhibitors

The table contains 136 products whose active ingredient are classified under the same pharmacologic class Breast Cancer Resistance Protein Inhibitors [MoA].

NDC Proprietary Name Non-Proprietary Name Dosage Form Route Name Company Name Status
0002-2980Retevmo Non-Proprietary Name: SelpercatinibCapsuleOralEli Lilly And CompanyACTIVE
0002-3977Retevmo Non-Proprietary Name: SelpercatinibCapsuleOralEli Lilly And CompanyACTIVE
0002-5340Retevmo Non-Proprietary Name: SelpercatinibTablet, CoatedOralEli Lilly And CompanyACTIVE
0002-5562Retevmo Non-Proprietary Name: SelpercatinibTablet, CoatedOralEli Lilly And CompanyACTIVE
0002-6082Retevmo Non-Proprietary Name: SelpercatinibTablet, CoatedOralEli Lilly And CompanyACTIVE
0002-6120Retevmo Non-Proprietary Name: SelpercatinibTablet, CoatedOralEli Lilly And CompanyACTIVE
0002-6902Jaypirca Non-Proprietary Name: PirtobrutinibTablet, CoatedOralEli Lilly And CompanyACTIVE
0002-7026Jaypirca Non-Proprietary Name: PirtobrutinibTablet, CoatedOralEli Lilly And CompanyACTIVE
0003-3641Evotaz Non-Proprietary Name: Atazanavir And CobicistatTabletOralE.r. Squibb & Sons, L.l.c.ACTIVE
0006-3074Zepatier Non-Proprietary Name: Elbasvir And GrazoprevirTablet, Film CoatedOralMerck Sharp & Dohme LlcACTIVE
0069-0227Lorbrena Non-Proprietary Name: LorlatinibTablet, Film CoatedOralPfizer Laboratories Div Pfizer IncACTIVE
0069-0231Lorbrena Non-Proprietary Name: LorlatinibTablet, Film CoatedOralPfizer Laboratories Div Pfizer IncACTIVE
0074-0522Kaletra Non-Proprietary Name: Lopinavir And RitonavirTablet, Film CoatedOralAbbvie Inc.ACTIVE
0074-2340Norvir Non-Proprietary Name: RitonavirTablet, Film CoatedOralAbbvie Inc.ACTIVE
0074-2600Mavyret Non-Proprietary Name: Glecaprevir And PibrentasvirPelletOralAbbvie Inc.ACTIVE
0074-2625Mavyret Non-Proprietary Name: Glecaprevir And PibrentasvirTablet, Film CoatedOralAbbvie Inc.ACTIVE
0074-3008Kaletra Non-Proprietary Name: Lopinavir And RitonavirTablet, Film CoatedOralAbbvie Inc.ACTIVE
0074-3399Norvir Non-Proprietary Name: RitonavirPowderOralAbbvie Inc.ACTIVE
0074-3956Kaletra Non-Proprietary Name: Lopinavir And RitonavirSolutionOralAbbvie Inc.ACTIVE
0074-4014Kaletra Non-Proprietary Name: Lopinavir And RitonavirTablet, Film CoatedOralAbbvie Inc.ACTIVE
0074-6799Kaletra Non-Proprietary Name: Lopinavir And RitonavirTablet, Film CoatedOralAbbvie Inc.ACTIVE
0078-0681Tafinlar Non-Proprietary Name: DabrafenibCapsuleOralNovartis Pharmaceuticals CorporationACTIVE
0078-0682Tafinlar Non-Proprietary Name: DabrafenibCapsuleOralNovartis Pharmaceuticals CorporationACTIVE
0078-0684Promacta Non-Proprietary Name: Eltrombopag OlamineTablet, Film CoatedOralNovartis Pharmaceuticals CorporationACTIVE
0078-0685Promacta Non-Proprietary Name: Eltrombopag OlamineTablet, Film CoatedOralNovartis Pharmaceuticals CorporationACTIVE
0078-0686Promacta Non-Proprietary Name: Eltrombopag OlamineTablet, Film CoatedOralNovartis Pharmaceuticals CorporationACTIVE
0078-0687Promacta Non-Proprietary Name: Eltrombopag OlamineTablet, Film CoatedOralNovartis Pharmaceuticals CorporationACTIVE
0078-0697Promacta Non-Proprietary Name: Eltrombopag OlaminePowder, For SuspensionOralNovartis Pharmaceuticals CorporationACTIVE
0078-0709Tabrecta Non-Proprietary Name: CapmatinibTablet, Film CoatedOralNovartis Pharmaceuticals CorporationACTIVE
0078-0716Tabrecta Non-Proprietary Name: CapmatinibTablet, Film CoatedOralNovartis Pharmaceuticals CorporationACTIVE
0078-0972Promacta Non-Proprietary Name: Eltrombopag OlaminePowder, For SuspensionOralNovartis Pharmaceuticals CorporationACTIVE
0078-1154Tafinlar Non-Proprietary Name: DabrafenibTablet, For SuspensionOralNovartis Pharmaceuticals CorporationACTIVE
0310-1349Tagrisso Non-Proprietary Name: OsimertinibTablet, Film CoatedOralAstrazeneca Pharmaceuticals LpACTIVE
0310-1350Tagrisso Non-Proprietary Name: OsimertinibTablet, Film CoatedOralAstrazeneca Pharmaceuticals LpACTIVE
0480-3273Alvaiz Non-Proprietary Name: EltrombopagTablet, Film CoatedOralTeva Pharmaceuticals, Inc.ACTIVE
0480-3274Alvaiz Non-Proprietary Name: EltrombopagTablet, Film CoatedOralTeva Pharmaceuticals, Inc.ACTIVE
0480-3275Alvaiz Non-Proprietary Name: EltrombopagTablet, Film CoatedOralTeva Pharmaceuticals, Inc.ACTIVE
0480-3276Alvaiz Non-Proprietary Name: EltrombopagTablet, Film CoatedOralTeva Pharmaceuticals, Inc.ACTIVE
0527-1947Lopinavir-ritonavir Non-Proprietary Name: Lopinavir-ritonavirSolutionOralLannett Company, Inc.ACTIVE
10147-0150Itraconazole Non-Proprietary Name: ItraconazoleSolutionOralPatriot Pharmaceuticals, LlcACTIVE
10147-1700Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralPatriot PharmaceuticalsACTIVE
13668-463Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralTorrent Pharmaceuticals LimitedACTIVE
16714-743Itraconazole Non-Proprietary Name: ItraconazoleCapsule, Coated PelletsOralNorthstar RxllcACTIVE
27505-110Xadago Non-Proprietary Name: Safinamide MesylateTablet, Film CoatedOralMdd Us Operations Llc, A Subsidiary Of Supernus Pharmaceuticals, Inc.ACTIVE
27505-111Xadago Non-Proprietary Name: Safinamide MesylateTablet, Film CoatedOralMdd Us Operations Llc, A Subsidiary Of Supernus Pharmaceuticals, Inc.ACTIVE
31722-006Itraconazole Non-Proprietary Name: ItraconazoleSolutionOralCamber Pharmaceuticals, Inc.ACTIVE
31722-045Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochlorideTabletOralCamber Pharmaceuticals, Inc.ACTIVE
31722-047Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralCamber Pharmaceuticals, Inc.ACTIVE
31722-048Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralCamber Pharmaceuticals, Inc.ACTIVE
31722-556Lopinavir And Ritonavir Non-Proprietary Name: Lopinavir And RitonavirTablet, Film CoatedOralCamber Pharmaceuticals, Inc.ACTIVE
31722-597Ritonavir Non-Proprietary Name: RitonavirTabletOralCamber Pharmaceuticals, Inc.ACTIVE
31722-603Lopinavir And Ritonavir Non-Proprietary Name: Lopinavir And RitonavirTablet, Film CoatedOralCamber Pharmaceuticals, Inc.ACTIVE
42385-933Lopinavir And Ritonavir Non-Proprietary Name: Lopinavir And RitonavirTablet, Film CoatedOralLaurus Labs LimitedACTIVE
42385-934Lopinavir And Ritonavir Non-Proprietary Name: Lopinavir And RitonavirTablet, Film CoatedOralLaurus Labs LimitedACTIVE
43598-096Javygtor Non-Proprietary Name: Sapropterin DihydrochlorideTabletOralDr. Reddys Laboratories IncACTIVE
43598-097Javygtor Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralDr. Reddys Laboratories IncACTIVE
43598-162Javygtor Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralDr. Reddys Laboratories IncACTIVE
43598-477Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralDr. Reddys Laboratories IncACTIVE
43598-749 Non-Proprietary Name: Sapropterin DihydrochlorideTabletDr. Reddy's Laboratories Inc.ACTIVE
43598-749Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochlorideTabletOralDr. Reddys Laboratories Inc.ACTIVE
46708-204Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralAlembic Pharmaceuticals LimitedACTIVE
49884-239Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralPar Pharmaceutical, Inc.ACTIVE
49884-720Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochlorideTabletOralPar Pharmaceutical, Inc.ACTIVE
49884-873Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralPar Pharmaceutical, Inc.ACTIVE
49884-948Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralPar Pharmaceutical, Inc.ACTIVE
50072-010Tpoxx Non-Proprietary Name: Tecovirimat MonohydrateInjection, Solution, ConcentrateIntravenousSiga Technologies, Inc.ACTIVE
50072-200Tpoxx Non-Proprietary Name: Tecovirimat MonohydrateCapsuleOralSiga Technologies, Inc.ACTIVE
50090-1723Prezcobix Non-Proprietary Name: Darunavir Ethanolate And CobicistatTablet, Film CoatedOralA-s Medication SolutionsACTIVE
50268-450Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralAvpakACTIVE
50419-171Stivarga Non-Proprietary Name: RegorafenibTablet, Film CoatedOralBayer Healthcare Pharmaceuticals Inc.ACTIVE
50458-290Sporanox Non-Proprietary Name: ItraconazoleCapsuleOralJanssen Pharmaceuticals, Inc.ACTIVE
50458-295Sporanox Non-Proprietary Name: ItraconazoleSolutionOralJanssen Pharmaceuticals, Inc.ACTIVE
51862-462Tolsura Non-Proprietary Name: ItraconazoleCapsule, Gelatin CoatedOralMayne Pharma Commercial LlcACTIVE
59676-575Prezcobix Non-Proprietary Name: Darunavir Ethanolate And CobicistatTablet, Film CoatedOralJanssen Products LpACTIVE
59676-800Symtuza Non-Proprietary Name: Darunavir, Cobicistat, Emtricitabine, And Tenofovir AlafenamideTablet, Film CoatedOralJanssen Products LpACTIVE
60687-299Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralAmerican Health PackagingACTIVE
60687-420Ritonavir Non-Proprietary Name: RitonavirTablet, Film CoatedOralAmerican Health PackagingACTIVE
61958-1201Stribild Non-Proprietary Name: Elvitegravir, Cobicistat, Emtricitabine, And Tenofovir Disoproxil FumarateTablet, Film CoatedOralGilead Sciences, Inc.ACTIVE
61958-1401Tybost Non-Proprietary Name: CobicistatTablet, Film CoatedOralGilead Sciences, Inc.ACTIVE
61958-1801Harvoni Non-Proprietary Name: Ledipasvir And SofosbuvirTablet, Film CoatedOralGilead Sciences, IncACTIVE
61958-1803Harvoni Non-Proprietary Name: Ledipasvir And SofosbuvirTablet, Film CoatedOralGilead Sciences, IncACTIVE
61958-1804Harvoni Non-Proprietary Name: Ledipasvir And SofosbuvirPelletOralGilead Sciences, IncACTIVE
61958-1805Harvoni Non-Proprietary Name: Ledipasvir And SofosbuvirPelletOralGilead Sciences, IncACTIVE
61958-1901Genvoya Non-Proprietary Name: Elvitegravir, Cobicistat, Emtricitabine, And Tenofovir AlafenamideTabletOralGilead Sciences, Inc.ACTIVE
61958-2201Epclusa Non-Proprietary Name: Velpatasvir And SofosbuvirTablet, Film CoatedOralGilead Sciences, Inc.ACTIVE
61958-2203Epclusa Non-Proprietary Name: Velpatasvir And SofosbuvirTablet, Film CoatedOralGilead Sciences, Inc.ACTIVE
61958-2204Epclusa Non-Proprietary Name: Velpatasvir And SofosbuvirPelletOralGilead Sciences, Inc.ACTIVE
61958-2205Epclusa Non-Proprietary Name: Velpatasvir And SofosbuvirPelletOralGilead Sciences, Inc.ACTIVE
61958-2401Vosevi Non-Proprietary Name: Sofosbuvir, Velpatasvir, And VoxilaprevirTablet, Film CoatedOralGilead Sciences, Inc.ACTIVE
62332-204Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralAlembic Pharmaceuticals Inc.ACTIVE
63539-927Lorbrena Non-Proprietary Name: LorlatinibTablet, Film CoatedOralU.s. PharmaceuticalsACTIVE
64764-800Livtencity Non-Proprietary Name: MaribavirTablet, CoatedOralTakeda Pharmaceuticals America, Inc.ACTIVE
64842-0120Lytgobi Non-Proprietary Name: FutibatinibTabletOralTaiho Pharmaceutical Co., Ltd.ACTIVE
65162-061Ritonavir Non-Proprietary Name: RitonavirTabletOralAmneal Pharmaceuticals LlcACTIVE
65162-087Itraconazole Non-Proprietary Name: ItraconazoleSolutionOralAmneal Pharmaceuticals LlcACTIVE
65162-630Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralAmneal Pharmaceuticals LlcACTIVE
65862-687 Non-Proprietary Name: RitonavirTablet, Film CoatedAurobindo Pharma LimitedACTIVE
65862-687Ritonavir Non-Proprietary Name: RitonavirTablet, Film CoatedOralAurobindo Pharma LimitedACTIVE
67877-454Itraconazole Non-Proprietary Name: ItraconazoleCapsule, Coated PelletsOralAscend Laboratories, LlcACTIVE
67919-040Sivextro Non-Proprietary Name: Tedizolid PhosphateInjection, Powder, Lyophilized, For SolutionIntravenousMerck Sharp & Dohme LlcACTIVE
67919-041Sivextro Non-Proprietary Name: Tedizolid PhosphateTablet, Film CoatedOralMerck Sharp & Dohme LlcACTIVE
68071-2348Kaletra Non-Proprietary Name: Lopinavir And RitonavirTablet, Film CoatedOralNucare Pharmaceuticals,inc.ACTIVE
68071-2949Lopinavir And Ritonavir Non-Proprietary Name: Lopinavir And RitonavirTablet, Film CoatedOralNucare Pharmaceuticals,inc.ACTIVE
68135-300Kuvan Non-Proprietary Name: Sapropterin DihydrochlorideTabletOralBiomarin Pharmaceutical Inc.ACTIVE
68135-301Kuvan Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralBiomarin Pharmaceutical Inc.ACTIVE
68135-482Kuvan Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralBiomarin Pharmaceutical Inc.ACTIVE
68382-697Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralZydus Pharmaceuticals Usa Inc.ACTIVE
69097-655Ritonavir film coatedNon-Proprietary Name: Ritonavir 100 MgTabletOralCipla Usa Inc.ACTIVE
69339-159Itraconazole Oral Non-Proprietary Name: ItraconazoleSolutionOralNatco Pharma Usa LlcACTIVE
69639-101Akynzeo Non-Proprietary Name: Netupitant And PalonosetronCapsuleOralHelsinn Therapeutics (u.s.), Inc.ACTIVE
70518-2872Itraconazole Non-Proprietary Name: ItraconazoleCapsule, Coated PelletsOralRemedyrepack Inc.ACTIVE
70518-3559Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralRemedyrepack Inc.ACTIVE
70720-101Varubi Non-Proprietary Name: RolapitantTabletOralTersera Therapeutics LlcACTIVE
70771-1208Itraconazole Non-Proprietary Name: ItraconazoleCapsuleOralZydus Lifesciences LimitedACTIVE
71274-170Joenja Non-Proprietary Name: LeniolisibTablet, Film CoatedOralPharming Healthcare Inc.ACTIVE
72000-310Sivextro Non-Proprietary Name: Tedizolid PhosphateTablet, Film CoatedOralNabriva Therapeutics Us, Inc.ACTIVE
72064-110Ayvakit Non-Proprietary Name: AvapritinibTablet, Film CoatedOralBlueprint Medicines CorporationACTIVE
72064-120Ayvakit Non-Proprietary Name: AvapritinibTablet, Film CoatedOralBlueprint Medicines CorporationACTIVE
72064-125Ayvakit Non-Proprietary Name: AvapritinibTablet, Film CoatedOralBlueprint Medicines CorporationACTIVE
72064-130Ayvakit Non-Proprietary Name: AvapritinibTablet, Film CoatedOralBlueprint Medicines CorporationACTIVE
72064-150Ayvakit Non-Proprietary Name: AvapritinibTablet, Film CoatedOralBlueprint Medicines CorporationACTIVE
72187-0101Orserdu Non-Proprietary Name: ElacestrantTablet, Film CoatedOralStemline Therapeutics, Inc.ACTIVE
72187-0102Orserdu Non-Proprietary Name: ElacestrantTablet, Film CoatedOralStemline Therapeutics, Inc.ACTIVE
72482-100Vonjo Non-Proprietary Name: PacritinibCapsuleOralCti Biopharma Corp.ACTIVE
72603-191Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochlorideTabletOralNorthstar RxllcACTIVE
72603-193Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralNorthstar RxllcACTIVE
72603-194Sapropterin Dihydrochloride Non-Proprietary Name: Sapropterin DihydrochloridePowder, For SolutionOralNorthstar RxllcACTIVE
72626-2601Ledipasvir And Sofosbuvir Non-Proprietary Name: Ledipasvir And SofosbuvirTablet, Film CoatedOralAsegua Therapeutics LlcACTIVE
72626-2701Sofosbuvir And Velpatasvir Non-Proprietary Name: Velpatasvir And SofosbuvirTablet, Film CoatedOralAsegua Therapeutics LlcACTIVE
72974-120 Non-Proprietary Name: RelugolixTablet, Film CoatedSumitomo Pharma America, Inc.ACTIVE
72974-120Orgovyx Non-Proprietary Name: RelugolixTablet, Film CoatedOralSumitomo Pharma America, IncACTIVE
72974-415Myfembree Non-Proprietary Name: Relugolix, Estradiol Hemihydrate, And Norethindrone AcetateTablet, Film CoatedOralSumitomo Pharma America, IncACTIVE
73079-050Zokinvy Non-Proprietary Name: LonafarnibCapsuleOralEiger Biopharmaceuticals, Inc.ACTIVE
73079-075Zokinvy Non-Proprietary Name: LonafarnibCapsuleOralEiger Biopharmaceuticals, Inc.ACTIVE
73207-101Qinlock Non-Proprietary Name: RipretinibTabletOralDeciphera Pharmaceuticals, LlcACTIVE